Synthesis and structure-activity relationships of carbohydrazides and 1,3,4-oxadiazole derivatives bearing an imidazolidine moiety against the yellow fever and dengue vector, Aedes aegypti

TOK F., Kocyigit-Kaymakcioglu B., Tabanca N., Estep A. S., Gross A. D., Geldenhuys W. J., ...Daha Fazla

PEST MANAGEMENT SCIENCE, cilt.74, sa.2, ss.413-421, 2018 (SCI-Expanded) identifier identifier identifier

  • Yayın Türü: Makale / Tam Makale
  • Cilt numarası: 74 Sayı: 2
  • Basım Tarihi: 2018
  • Doi Numarası: 10.1002/ps.4722
  • Dergi Adı: PEST MANAGEMENT SCIENCE
  • Derginin Tarandığı İndeksler: Science Citation Index Expanded (SCI-EXPANDED), Scopus
  • Sayfa Sayıları: ss.413-421
  • Anahtar Kelimeler: insecticide, mosquitocidal activity, mosquito control, carbohydrazide and amide, mitochondria, INSECTICIDAL ACTIVITY, DESIGN, ANTICANCER, INHIBITORS, OXADIAZOLE, AGENTS, RINGS, MODE
  • Marmara Üniversitesi Adresli: Evet

Özet

BACKGROUND 1,3,4-Oxadiazole and imidazolidine rings are important heterocyclic compounds exhibiting a variety of biological activities. In this study, novel compounds with oxadiazole and imidazolidine rings were synthesized from 3-(methylsulfonyl)-2-oxoimidazolidine-1-carbonyl chloride and screened for insecticidal activities. The proposed structures of the 17 synthesized compounds were confirmed using elemental analysis, infrared (IR), proton nuclear magnetic resonance (H-1-NMR), and mass spectroscopy.